SCHEMBL18399147

SCHEMBL18399147

Cc1cc2cn[nH]c2cc1OC(=O)N1CCNCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AXL P30530 1/20 0.38
MKNK1 Q9BUB5 3/20 0.38
TRPV1 Q8NER1 4/20 0.37
ROCK2 O75116 3/20 0.36
CYP3A4 P08684 2/20 0.36
BTK Q06187 2/20 0.35
LCK P06239 1/20 0.35
LYN P07948 1/20 0.35
HCK P08631 1/20 0.35
FGR P09769 1/20 0.35
SRC P12931 1/20 0.35
TEC P42680 1/20 0.35
FRK P42685 1/20 0.35
BLK P51451 1/20 0.35
BMX P51813 1/20 0.35
LIMK1 P53667 1/20 0.35
ACVR1 Q04771 1/20 0.35
TNK2 Q07912 1/20 0.35
ITK Q08881 1/20 0.35
ACACB O00763 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18399006 0.89 MKNK1 (0.46) AXLMKNK1ROCK2CYP3A4L3MBTL1
SCHEMBL18399106 0.87 TSHR (0.47)
SCHEMBL18399071 0.78 SMN1; SMN2 (0.48) TRPV1L3MBTL1
SCHEMBL18399231 0.75 CHEK1 (0.40) LIMK1
SCHEMBL18399204 0.74 TDP1 (0.45) MKNK1ROCK2L3MBTL1
SCHEMBL25313919 0.73 GABRP (0.40)
SCHEMBL31721821 0.72 ALDH1A1 (0.50) AXLTRPV1ROCK2CYP3A4BTK
SCHEMBL22750070 0.71 ROCK2 (0.47) ROCK2PDGFRBPDGFRA
SCHEMBL25258769 0.70 SMN1; SMN2 (0.52) CYP3A4
SCHEMBL20617830 0.69 AXL (0.67) AXLMKNK1TRPV1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3325449-A1 COMPOUNDS GlaxoSmithKline Intellectual Property Development Limited (GB) 2018-05-30 EP disclosed
WO-2017012576-A1 COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-01-26 WO disclosed