SCHEMBL1840370

SCHEMBL1840370

CCOC(=O)C(C)(C)Oc1ccc(OCC(C2CCCCC2)C2(c3ccc(Cl)cc3)Nc3cc(F)c(F)cc3N2)c(C)c1C

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
TSHR P16473 1/20 0.37
HTR2A P28223 1/20 0.37
PMP22 Q01453 1/20 0.37
PPARA Q07869 1/20 0.37
FBP1 P09467 6/20 0.35
LMNA P02545 1/20 0.33
HSD11B1 P28845 1/20 0.32
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1841851 0.92 PTGDR2 (0.33) CYP1A2CYP3A4PPARALMNAMAPT
SCHEMBL200871 0.91 PPARA (0.42) ABCB11CYP1A2CYP3A4TSHRHTR2A
SCHEMBL1842335 0.89 PPARA (0.47) ABCB11CYP1A2CYP3A4TSHRHTR2A
SCHEMBL1839730 0.87 PPARA (0.41) ABCB11CYP1A2CYP3A4TSHRHTR2A
SCHEMBL198730 0.85 PPARA (0.41) ABCB11CYP1A2CYP3A4TSHRHTR2A
SCHEMBL1843200 0.81 PPARA (0.37) CYP1A2CYP3A4PPARAMAPT
SCHEMBL1838605 0.81 ALOX15 (0.37) TSHR
SCHEMBL1841206 0.80 HPD (0.37)
SCHEMBL198388 0.80 PPARA (0.42) CYP1A2CYP3A4TSHRPPARALMNA
SCHEMBL1837083 0.80 GAA (0.39) LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2321282-A1 NEW BENZIMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2011-05-18 EP disclosed
WO-2010028981-A1 NEW BENZIMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-03-18 WO disclosed