SCHEMBL1840448

SCHEMBL1840448

N=C(N)N(C(=O)OCc1ccccc1)C(=O)c1ccc(C2=CCN(C(=O)O)CC2)c(C(F)(F)F)c1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 7/20 0.38
MMP2 P08253 1/20 0.36
MMP3 P08254 1/20 0.36
LNPEP Q9UIQ6 1/20 0.35
BTK Q06187 2/20 0.34
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
MAPT P10636 1/20 0.33
MTOR P42345 1/20 0.33
TRPV1 Q8NER1 2/20 0.33
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
HPN P05981 1/20 0.32
ST14 Q9Y5Y6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1763979 0.91 PDK4 (0.42) PTGDR2LNPEPBTK
SCHEMBL1763543 0.74 ADH5 (0.41) MMP2MMP3MAPTTRPV1PPARG
SCHEMBL1840656 0.72 NOTUM (0.44) MMP2MMP3MAPTTRPV1
SCHEMBL2040083 0.70 PTGDR2 (0.54) PTGDR2LNPEP
SCHEMBL1763851 0.70 SLC9A1 (0.45)
SCHEMBL28909629 0.70 TSHR (0.46) MMP2MMP3MAPTMTORTRPV1
SCHEMBL3325476 0.70 MAPT (0.50) MMP2MMP3JAK1MAPTTRPV1
SCHEMBL23777377 0.70 KMT2A (0.50) MAPT
SCHEMBL2037929 0.69 PTGDR2 (0.54) PTGDR2LNPEP
SCHEMBL1763602 0.69 P2RX7 (0.39) PTGDR2MMP2MMP3BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2321274-A1 PYRROLIDINYL AND PIPERIDINYL COMPOUNDS USEFUL AS NHE-1 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2011-05-18 EP disclosed
WO-2010005783-A1 PYRROLIDINYL AND PIPERIDINYL COMPOUNDS USEFUL AS NHE-1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-01-14 WO disclosed