SCHEMBL18404686

SCHEMBL18404686

COC(=O)CC(NC(=O)CN)c1ccc(O)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.43
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
TACR3 P29371 1/20 0.38
RAB9A P51151 2/20 0.37
MAPT P10636 2/20 0.37
HTT P42858 2/20 0.36
ALDH1A1 P00352 2/20 0.36
LMNA P02545 1/20 0.36
TAAR1 Q96RJ0 2/20 0.35
HTR3A P46098 1/20 0.35
TSHR P16473 1/20 0.35
NFKB1 P19838 1/20 0.35
HIF1A Q16665 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18404162 0.87 ALDH1A1 (0.50) POLBKMT2AMEN1SMN1; SMN2MAPT
SCHEMBL6668682 0.85 ALDH1A1 (0.46) POLBKMT2AMEN1SMN1; SMN2MAPT
SCHEMBL6667674 0.85 MEN1 (0.51) POLBKMT2AMEN1SMN1; SMN2TACR3
SCHEMBL6671131 0.83 POLB (0.47) POLBKMT2AMEN1MAPT
SCHEMBL6668894 0.83 HTT (0.47) POLBKMT2AMEN1TACR3MAPT
SCHEMBL24036553 0.83 THRB (0.47) POLBKMT2AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL7176606 0.83 MEN1 (0.50) POLBKMT2AMEN1SMN1; SMN2TACR3
SCHEMBL7365092 0.82 ALDH1A1 (0.50) KMT2AMEN1MAPTHTTALDH1A1
Hydrochloric Acid SCHEMBL7176273 0.82 POLB (0.46) POLBKMT2AMAPT
Hydrochloric Acid SCHEMBL7170943 0.82 HTT (0.46) POLBKMT2AMEN1TACR3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2534138-B1 1,2,3-TRIAZOLE-BASED PEPTIDOMIMETIC INTEGRIN INHIBITORS FOR THE DIAGNOSIS AND THERAPY OF TUMORS UNIVERSITA' DEGLI STUDI DI FIRENZE (IT) 2017-01-25 EP disclosed