SCHEMBL18408249

SCHEMBL18408249

CC1C2Cc3ccc(-c4ccc(=O)n(C)n4)cc3[C@]1(C)CCN2

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.55
OPRD1 P41143 3/20 0.55
OPRK1 P41145 3/20 0.55
SIGMAR1 Q99720 3/20 0.55
HRH3 Q9Y5N1 12/20 0.43
MRGPRX2 Q96LB1 2/20 0.40
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1207194 1.00 OPRM1 (0.55) OPRM1OPRD1OPRK1SIGMAR1HRH3
SCHEMBL18408255 0.83 OPRM1 (0.57) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL1207863 0.83 OPRM1 (0.57) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL1206851 0.81 OPRM1 (0.57) OPRM1OPRD1OPRK1SIGMAR1HRH3
SCHEMBL18408049 0.81 OPRM1 (0.57) OPRM1OPRD1OPRK1SIGMAR1HRH3
SCHEMBL18408180 0.78 OPRM1 (0.59) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL1206692 0.78 OPRM1 (0.59) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL2582641 0.78 OPRM1 (0.59) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL1207662 0.76 OPRD1 (0.63) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2
SCHEMBL18407995 0.76 OPRD1 (0.63) OPRM1OPRD1OPRK1SIGMAR1MRGPRX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2220048-B1 ARYL- AND HETEROARYLCARBONYL DERIVATIVES OF BENZOMORPHANES AND RELATED SCAFFOLDS, MEDICAMENTS CONTAINING SUCH COMPOUNDS AND THEIR USE BOEHRINGER INGELHEIM INT (DE) 2017-01-25 EP disclosed