SCHEMBL18409702

SCHEMBL18409702

Fc1ccc(-c2nc(CCCc3c[nH]c4ccccc34)oc2-c2ccc(F)c(-c3cc(Cl)cc(-c4nc(CCCc5c[nH]c6ccccc56)oc4-c4cccc(Cl)c4)c3)c2)cc1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.43
RXRA P19793 8/20 0.43
RXRB P28702 8/20 0.43
RXRG P48443 8/20 0.43
NR4A2 P43354 1/20 0.43
GPR84 Q9NQS5 1/20 0.39
NAMPT P43490 1/20 0.38
HTR1A P08908 1/20 0.35
PTPN1 P18031 1/20 0.35
CDK4 P11802 1/20 0.35
CCND1 P24385 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18409657 0.90 RXRA (0.41) HTR6RXRARXRBRXRGNR4A2
SCHEMBL18409643 0.85 HTR6 (0.54) HTR6RXRARXRBRXRGNR4A2
SCHEMBL18409639 0.83 GPR84 (0.52) RXRARXRBRXRGNR4A2GPR84
SCHEMBL18409637 0.80 CDK4 (0.46) HTR6RXRARXRBRXRGGPR84
SCHEMBL22692981 0.77 NR4A2 (0.46) HTR6RXRARXRBRXRGNR4A2
SCHEMBL18409642 0.77 NR4A2 (0.53) HTR6RXRARXRBRXRGNR4A2
SCHEMBL18409339 0.75 HTR6 (0.52) HTR6RXRARXRBRXRGNR4A2
SCHEMBL18409633 0.75 PTPN1 (0.45) HTR6RXRARXRBRXRGNR4A2
SCHEMBL18409641 0.74 CDK4 (0.47) HTR6RXRARXRBRXRGGPR84
SCHEMBL18409723 0.74 RXRA (0.54) HTR6RXRARXRBRXRGPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017011920-A1 COMPOUNDS AND USES THEREOF IN THE TREATMENT OF CANCERS AND OTHER MEDICAL CONDITIONS THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING/MCGILL UNIVERSITY (CA) 2017-01-26 WO disclosed