SCHEMBL18436755

SCHEMBL18436755

Bc1ccc(N2C[C@@H](C)O[C@@H](C)C2)nc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.51
AOC3 Q16853 3/20 0.41
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 2/20 0.41
RAB9A P51151 1/20 0.41
GAA P10253 1/20 0.41
ADRA1A P35348 1/20 0.40
TLR9 Q9NR96 1/20 0.40
TLR8 Q9NR97 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
MAP3K12 Q12852 1/20 0.40
TDP1 Q9NUW8 2/20 0.40
HPGD P15428 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HTT P42858 1/20 0.38
ACVR1 Q04771 1/20 0.38
LMNA P02545 1/20 0.37
MAP3K7 O43318 2/20 0.37
PIK3CA P42336 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10034110 0.81 KMT2A (0.53) KMT2AAOC3KDM4EALDH1A1MAPT
SCHEMBL24018507 0.81 KMT2A (0.53) KMT2AAOC3KDM4EALDH1A1MAPT
SCHEMBL18436130 0.81 KMT2A (0.53) KMT2AAOC3KDM4EALDH1A1MAPT
SCHEMBL15743968 0.81 KMT2A (0.53) KMT2AAOC3KDM4EALDH1A1MAPT
SCHEMBL31182223 0.81 KMT2A (0.53) KMT2AAOC3KDM4EALDH1A1MAPT
SCHEMBL20456804 0.80 KMT2A (0.51) KMT2AAOC3KDM4EALDH1A1MAPT
SCHEMBL17803130 0.80 KMT2A (0.51) KMT2AAOC3KDM4EALDH1A1MAPT
SCHEMBL18307179 0.80 KMT2A (0.51) KMT2AAOC3KDM4EALDH1A1MAPT
SCHEMBL20004006 0.80 KMT2A (0.51) KMT2AAOC3KDM4EALDH1A1MAPT
SCHEMBL23019809 0.80 KMT2A (0.51) KMT2AAOC3KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-B1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO LTD (CN) 2019-09-11 EP disclosed
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed