SCHEMBL18307179

SCHEMBL18307179

CC1CN(c2ccc(I)cn2)CC(C)O1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.51
AOC3 Q16853 3/20 0.41
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 2/20 0.41
RAB9A P51151 2/20 0.41
MAPT P10636 2/20 0.41
ADRA1A P35348 1/20 0.40
TLR9 Q9NR96 1/20 0.40
TLR8 Q9NR97 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
TDP1 Q9NUW8 2/20 0.40
HPGD P15428 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.38
NPC1 O15118 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ACVR1 Q04771 1/20 0.38
MAP3K12 Q12852 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20456804 1.00 KMT2A (0.51) KMT2AAOC3KDM4EALDH1A1GAA
SCHEMBL10034110 0.81 KMT2A (0.53) KMT2AAOC3KDM4EALDH1A1GAA
SCHEMBL18436130 0.81 KMT2A (0.53) KMT2AAOC3KDM4EALDH1A1GAA
SCHEMBL31182223 0.81 KMT2A (0.53) KMT2AAOC3KDM4EALDH1A1GAA
SCHEMBL15743968 0.81 KMT2A (0.53) KMT2AAOC3KDM4EALDH1A1GAA
SCHEMBL24018507 0.81 KMT2A (0.53) KMT2AAOC3KDM4EALDH1A1GAA
SCHEMBL20456715 0.80 MAP3K12 (0.38) MAP3K12PIK3CAMTOR
SCHEMBL18436755 0.80 KMT2A (0.51) KMT2AAOC3KDM4EALDH1A1GAA
SCHEMBL22837868 0.80 SORD (0.35) MAPT
SCHEMBL1080321 0.80 KMT2A (0.51) KMT2AAOC3KDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2265607-B1 PYRIMIDINE-2-AMINE COMPOUNDS AND THEIR USE AS INHIBITORS OF JAK KINASES RIGEL PHARMACEUTICALS INC (US) 2016-12-14 EP disclosed