SCHEMBL18436757

SCHEMBL18436757

Cc1cnc2c(-c3ccc(C#N)cc3)cccc2c1C1CC1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.43
CYP11B2 P19099 11/20 0.37
KDM1A O60341 4/20 0.37
CYP11B1 P15538 8/20 0.37
MAOB P27338 1/20 0.35
AKT1 P31749 1/20 0.35
KDM4A O75164 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
LAP3 P28838 1/20 0.34
PRKDC P78527 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21336962 0.82 HRH4 (0.40) HRH4CYP11B2KDM1AKDM4AKDM5B
SCHEMBL17128231 0.81 BRS3 (0.45) HRH4CYP11B2CYP11B1KDM4AKDM5B
SCHEMBL17128238 0.80 PDE5A (0.44) CYP11B2CYP11B1
SCHEMBL18436887 0.79 HRH4 (0.42) HRH4KDM1APRKDC
SCHEMBL17127884 0.79 HRH4 (0.42) HRH4KDM1APRKDC
SCHEMBL17128081 0.79 HRH4 (0.43) HRH4KDM1AMAOBPRKDC
SCHEMBL18436763 0.78 HRH4 (0.38) HRH4CYP11B2KDM1ACYP11B1MAOB
SCHEMBL21336710 0.78 HRH4 (0.40) HRH4CYP11B2CYP11B1KDM4AKDM5B
SCHEMBL17128328 0.77 HRH4 (0.42) HRH4CYP11B2KDM1ACYP11B1KDM4A
SCHEMBL17127837 0.77 HRH4 (0.40) HRH4KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed