SCHEMBL18436763

SCHEMBL18436763

N#Cc1ccc(-c2cccc3c(C4CC4)c(NCCN)cnc23)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.38
ACP1 P24666 1/20 0.34
KDM4A O75164 1/20 0.33
KDM5B Q9UGL1 1/20 0.33
KDM1A O60341 4/20 0.32
LAP3 P28838 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
FERMT2 Q96AC1 1/20 0.32
CA12 O43570 1/20 0.32
CA3 P07451 1/20 0.32
CA4 P22748 1/20 0.32
CA6 P23280 1/20 0.32
CA5A P35218 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
CA14 Q9ULX7 1/20 0.32
CA5B Q9Y2D0 1/20 0.32
SRC P12931 1/20 0.32
CCNA2 P20248 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21336647 0.82 KDM1A (0.36) HRH4KDM1ASRCCCNA2CDK2
SCHEMBL21336936 0.81 PDE9A (0.34) HRH4ACP1KDM1A
SCHEMBL18436916 0.81 DPP4 (0.34) HRH4KDM1ACCNA2CDK2
SCHEMBL18436682 0.80 RAD52 (0.38) HRH4ACP1KDM4AKDM5BKDM1A
SCHEMBL18436897 0.79 KDM4A (0.36) HRH4KDM4AKDM5BCYP11B1CYP11B2
SCHEMBL18436757 0.78 HRH4 (0.43) HRH4KDM4AKDM5BKDM1ALAP3
SCHEMBL17128231 0.74 BRS3 (0.45) HRH4KDM4AKDM5BLAP3CYP11B1
SCHEMBL18436776 0.72 HRH4 (0.35) HRH4CYP11B1CYP11B2CCNA2CDK2
SCHEMBL17128081 0.72 HRH4 (0.43) HRH4KDM1AMAOBMAPT
SCHEMBL21336962 0.71 HRH4 (0.40) HRH4KDM4AKDM5BKDM1ACYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed