SCHEMBL18436897

SCHEMBL18436897

CS(=O)(=O)CCC(=O)NCCNc1cnc2c(-c3ccc(C#N)cc3)cccc2c1C1CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4A O75164 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
CYP11B2 P19099 9/20 0.34
CYP11B1 P15538 7/20 0.34
SLC22A12 Q96S37 1/20 0.34
HRH4 Q9H3N8 1/20 0.33
CNR2 P34972 1/20 0.33
CCNT1 O60563 1/20 0.32
CCNK O75909 1/20 0.32
CCNA2 P20248 1/20 0.32
CDK2 P24941 1/20 0.32
CDK9 P50750 1/20 0.32
CDK12 Q9NYV4 1/20 0.32
HTR1A P08908 2/20 0.31
DRD2 P14416 2/20 0.31
HTR7 P34969 2/20 0.31
HTR6 P50406 2/20 0.31
HSD11B1 P28845 1/20 0.31
FLT3 P36888 1/20 0.31
EGLN1 Q9GZT9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18420199 0.81 KDM4A (0.40) KDM4AKDM5BCYP11B2CYP11B1SLC22A12
SCHEMBL18436763 0.79 HRH4 (0.38) KDM4AKDM5BCYP11B2CYP11B1HRH4
SCHEMBL17127865 0.78 RET (0.41) HRH4HTR1ADRD2HTR7HTR6
SCHEMBL18436916 0.76 DPP4 (0.34) HRH4CCNT1CCNKCCNA2CDK2
SCHEMBL21336647 0.76 KDM1A (0.36) HRH4CCNA2CDK2
SCHEMBL21336936 0.75 PDE9A (0.34) HRH4
SCHEMBL18436930 0.73 POLB (0.39) KDM4AKDM5BCYP11B2CYP11B1CNR2
SCHEMBL18436545 0.73 MTNR1A (0.39) KDM4AKDM5BCYP11B2CYP11B1CNR2
SCHEMBL21336770 0.72 EGLN1 (0.40) EGLN1
SCHEMBL17128231 0.71 BRS3 (0.45) KDM4AKDM5BCYP11B2CYP11B1SLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed