SCHEMBL184434

SCHEMBL184434

[C]1=COc2ccccc2O1

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 1/20 0.32
ITGB2 P05107 1/20 0.32
ICAM1 P05362 1/20 0.32
ITGAL P20701 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17288933 0.69 ADAMTS4 (0.32)
SCHEMBL17289186 0.69
SCHEMBL7172036 0.67 ABCG2 (0.40) ABCG2ITGB2ICAM1ITGAL
SCHEMBL452883 0.67
SCHEMBL17289110 0.66 CA1 (0.38) ABCG2
SCHEMBL451675 0.65 TRPA1 (0.30)
SCHEMBL17289161 0.65 TRPA1 (0.40)
SCHEMBL3557 0.64
SCHEMBL121647 0.64 LMNA (0.43) ABCG2ITGB2ICAM1ITGAL
SCHEMBL30334802 0.64 LMNA (0.43) ABCG2ITGB2ICAM1ITGAL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1390 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023237097-A1 19-NOR-C3,3-DISUBSTITUTED C21-AZACYCLO-SUBSTITUTED STEROID AND METHOD FOR USING SAME 山东绿叶制药有限公司 2023-12-14 WO claimed
EP-3409668-B1 NOVEL IMIDAZOLE DERIVATIVE HAVING JNK INHIBITORY ACTIVITY AND USE THEREOF SAMJIN PHARM CO LTD (KR) 2020-10-21 EP claimed
US-10781201-B2 Benzimidazole derivative having JNK inhibitory activity and use thereof INDUSTRY-UNIVERSITY COOPERATION FOUNDATION HANYANG UNIVERSITY ERICA CAMPUS (KR) 2020-09-22 US claimed
US-20200039959-A1 NOVEL BENZIMIDAZOLE DERIVATIVE HAVING JNK INHIBITORY ACTIVITY AND USE THEREOF INDUSTRY-UNIVERSITY COOPERATION FOUNDATION HANYANG UNIVERSITY ERICA CAMPUS (KR) 2020-02-06 US claimed
EP-3242872-B1 (PIPERIDIN-3-YL)(NAPHTHALEN-2-YL)METHANONE DERIVATIVES AND RELATED COMPOUNDS AS INHIBITORS OF THE HISTONE DEMETHYLASE KDM2B FOR THE TREATMENT OF CANCER GENENTECH INC (US) 2019-07-03 EP claimed
EP-3010906-B1 BENZIMIDAZOLE DERIVATIVES AS SELECTIVE PROTEIN KINASE INHIBITORS AB SCIENCE (FR) 2019-06-12 EP claimed
US-10301291-B2 Imidazole derivative having JNK inhibitory activity and use thereof SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2019-05-28 US claimed
US-10280149-B2 Therapeutic compounds and uses thereof GENENTECH, INC. (US) 2019-05-07 US claimed
US-20190031645-A1 NOVEL IMIDAZOLE DERIVATIVE HAVING JNK INHIBITORY ACTIVITY AND USE THEREOF INDUSTRY-UNIVERSITY COOPERATION FOUNDATION HANYANG UNIVERSITY ERICA CAMPUS (KR) 2019-01-31 US claimed
EP-3409668-A1 NOVEL IMIDAZOLE DERIVATIVE HAVING JNK INHIBITORY ACTIVITY AND USE THEREOF Samjin Pharmaceutical Co., Ltd. (KR) 2018-12-05 EP claimed
US-5804586-A ANALGESICS, PSYCHOLOGICAL DISORDERS KNOLL AKTIENGESELLSCHAFT (DE) 1998-09-08 US claimed
WO-1998018757-A1 SYNTHESIS OF BENZO[F]QUINOLINONES ELI LILLY AND COMPANY (US) 1998-05-07 WO claimed
EP-0707570-B1 ISOQUINOLINE DERIVATIVES AS THERAPEUTIC AGENTS KNOLL AG (DE) 1998-05-06 EP claimed
EP-0839807-A1 Synthesis of benzo(f)quinolinones ELI LILLY AND COMPANY (US) 1998-05-06 EP claimed
EP-0707570-A1 ISOQUINOLINE DERIVATIVES AS THERAPEUTIC AGENTS Knoll AG (DE) 1996-04-24 EP claimed
EP-0656885-A1 SYNTHESIS OF 2-SUBSTITUTED QUINAZOLINE COMPOUNDS (SUCH AS TERAZOSIN) AND MEOBENTINE AND BETHANIDINE AND INTERMEDIATES THEREFOR ACIC (CANADA) INC. (CA) 1995-06-14 EP claimed
WO-1995000489-A1 ISOQUINOLINE DERIVATIVES AS THERAPEUTIC AGENTS KNOLL AG (DE) 1995-01-05 WO claimed
WO-1994005628-A1 SYNTHESIS OF 2-SUBSTITUTED QUINAZOLINE COMPOUNDS (SUCH AS TERAZOSIN) AND MEOBENTINE AND BETHANIDINE AND INTERMEDIATES THEREFOR ACIC (CANADA) INC. (CA) 1994-03-17 WO claimed
EP-0114850-B1 NEW SUBSTITUTED DERIVATIVES OF 2,5-DIAMINO 1,4-DIAZOLE, PREPARATION METHODS THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BOUCHARA S.A. (FR) 1988-06-29 EP claimed
US-4569933-A Antihypertensive substituted derivatives of 2,5-diamino 1,4-diazole CORNU PIERRE JEAN 1986-02-11 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190031645-A1 NOVEL IMIDAZOLE DERIVATIVE HAVING JNK INHIBITORY ACTIVITY AND USE THEREOF MAPKAPK2, MAPKAPK3, MAP3K7 ABCG2 2469/4885ITGB2 4768/4885ICAM1 1380/4885
US-10301291-B2 Imidazole derivative having JNK inhibitory activity and use thereof MAPKAPK2, MAPKAPK3, MAP3K7 ABCG2 2305/4885ITGB2 4776/4885ICAM1 1073/4885
US-10280149-B2 Therapeutic compounds and uses thereof KDM1B, KDM6B, KDM2B ABCG2 4006/4885ITGB2 3670/4885ICAM1 3260/4885
US-20200039959-A1 NOVEL BENZIMIDAZOLE DERIVATIVE HAVING JNK INHIBITORY ACTIVITY AND USE THEREOF MAPKAPK3, MAPK3, MAP3K3 ABCG2 2556/4885ITGB2 4649/4885ICAM1 2478/4885
US-10781201-B2 Benzimidazole derivative having JNK inhibitory activity and use thereof MAPKAPK3, MAPK3, MAP3K3 ABCG2 2298/4885ITGB2 4623/4885ICAM1 2789/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.