SCHEMBL18456151

SCHEMBL18456151

CC1(C)c2ccccc2-c2c(-c3nc(-c4ccccc4)nc4ccc(-c5cccc6c5-c5ccccc5C65c6ccccc6-c6ccccc65)cc34)cccc21

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
WHR1 P49842 1/20 0.36
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ATM Q13315 1/20 0.33
NPC1 O15118 1/20 0.32
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32
NT5E P21589 1/20 0.30
TRIM58 Q8NG06 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18456117 0.89 ATM (0.40) MEN1KMT2AATMNPC1HTT
SCHEMBL18456152 0.89 WHR1 (0.43) WHR1MEN1KMT2AATMNPC1
SCHEMBL18455594 0.88 WHR1 (0.42) WHR1MEN1KMT2AATMNPC1
SCHEMBL18456157 0.83 WHR1 (0.41) WHR1MEN1KMT2AATMNT5E
SCHEMBL18456034 0.83 MEN1 (0.46) WHR1MEN1KMT2AATMNPC1
SCHEMBL18456041 0.82 WHR1 (0.44) WHR1MEN1KMT2AATM
SCHEMBL18456030 0.82 ADORA2A (0.36) MEN1KMT2AATMMAPK1
SCHEMBL20465240 0.82 MEN1 (0.35) MEN1KMT2A
SCHEMBL18456318 0.81 MEN1 (0.47) MEN1KMT2AATM
SCHEMBL23936024 0.81 WHR1 (0.45) WHR1MEN1KMT2AATMNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11201296-B2 Compounds having fluorene structures MERCK PATENT GMBH (DE) 2021-12-14 US disclosed
EP-3328850-B1 COMPOUNDS HAVING FLUORENE STRUCTURES MERCK PATENT GMBH (DE) 2020-11-11 EP disclosed
US-20180226587-A1 COMPOUNDS HAVING FLUORENE STRUCTURES MERCK PATENT GMBH (DE) 2018-08-09 US disclosed
US-20180226587-A1 COMPOUNDS HAVING FLUORENE STRUCTURES MERCK PATENT GMBH (DE) 2018-08-09 US disclosed
WO-2017016667-A1 COMPOUNDS HAVING FLUORENE STRUCTURES MERCK PATENT GMBH (DE) 2017-02-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180226587-A1 COMPOUNDS HAVING FLUORENE STRUCTURES FSCN1, EFNA1, FLNA WHR1 4335/4885MEN1 1658/4885KMT2A 2095/4885
US-11201296-B2 Compounds having fluorene structures FSCN1, EFNA1, FLNA WHR1 4335/4885MEN1 1658/4885KMT2A 2095/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.