SCHEMBL18458029

SCHEMBL18458029

CCC(O)N(CC1(N2CCN(Cc3ccccc3)CC2)CCOC(C)(C)C1)c1cccc(C#N)n1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 19/20 0.55
OPRM1 P35372 18/20 0.55
KCNH2 Q12809 9/20 0.55
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HIF1A Q16665 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18425607 0.85 SIGMAR1 (0.76) SIGMAR1OPRM1KCNH2
SCHEMBL18458560 0.78 OPRM1 (0.52) SIGMAR1OPRM1KCNH2
SCHEMBL21337259 0.78 OPRM1 (0.39) SIGMAR1OPRM1KCNH2
SCHEMBL18458529 0.77 OPRM1 (0.47) SIGMAR1OPRM1KCNH2ALDH1A1LMNA
SCHEMBL21337382 0.77 OPRM1 (0.43) SIGMAR1OPRM1KCNH2
SCHEMBL20621716 0.77 SIGMAR1 (0.48) SIGMAR1OPRM1KCNH2
SCHEMBL18423973 0.75 OPRM1 (0.48) SIGMAR1OPRM1KCNH2ALDH1A1LMNA
SCHEMBL18458556 0.75 SIGMAR1 (0.71) SIGMAR1OPRM1KCNH2
SCHEMBL19631818 0.74 SIGMAR1 (0.54) SIGMAR1OPRM1KCNH2LMNA
SCHEMBL18458564 0.74 OPRM1 (0.60) SIGMAR1OPRM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017016669-A1 SUBSTITUTED AMIDE DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2017-02-02 WO disclosed