SCHEMBL18458552

SCHEMBL18458552

CCC1OC1N(CC1(N2CCN(CCC(C)C)CC2)CCOCC1)c1cccc(C#N)n1

nearest known ligand 0.40

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 19/20 0.40
SIGMAR1 Q99720 19/20 0.40
KCNH2 Q12809 7/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18458562 0.82 OPRM1 (0.39) OPRM1SIGMAR1KCNH2
SCHEMBL21337382 0.81 OPRM1 (0.43) OPRM1SIGMAR1KCNH2
SCHEMBL18425965 0.81 OPRM1 (0.62) OPRM1SIGMAR1KCNH2
SCHEMBL21327078 0.77 OPRM1 (0.36) OPRM1SIGMAR1KCNH2
SCHEMBL18458374 0.74 OPRM1 (0.35) OPRM1SIGMAR1KCNH2
SCHEMBL18458560 0.73 OPRM1 (0.52) OPRM1SIGMAR1KCNH2
SCHEMBL18458551 0.72 OPRM1 (0.73) OPRM1SIGMAR1KCNH2
SCHEMBL21337556 0.72 SIGMAR1 (0.67) OPRM1SIGMAR1KCNH2
SCHEMBL21337259 0.71 OPRM1 (0.39) OPRM1SIGMAR1KCNH2
SCHEMBL18458558 0.71 OPRM1 (0.58) OPRM1SIGMAR1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017016669-A1 SUBSTITUTED AMIDE DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2017-02-02 WO disclosed