SCHEMBL1847685

SCHEMBL1847685

CC(O)(c1cccc(C(F)(F)F)c1)c1cc2cccc(-c3cccc(C(=O)O)c3)c2s1.CC(O)(c1cccc(C(F)(F)F)c1)c1cc2cccc(-c3cccc(C(N)=O)c3)c2s1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 6/20 0.47
S1PR4 O95977 1/20 0.43
S1PR5 Q9H228 1/20 0.43
DHODH Q02127 2/20 0.41
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
AKR1C3 P42330 2/20 0.38
AKR1C2 P52895 2/20 0.38
CFTR P13569 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
PLG P00747 1/20 0.37
PLAU P00749 1/20 0.37
PLAT P00750 1/20 0.37
PDE4A P27815 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3215806 0.96 GPR52 (0.50) GPR52S1PR4S1PR5DHODHAKR1C3
SCHEMBL3209033 0.95 GPR52 (0.47) GPR52S1PR4S1PR5RXRARXRB
SCHEMBL1847676 0.88 GPR52 (0.44) GPR52S1PR4S1PR5ALDH1A1AKR1C3
SCHEMBL1851681 0.84 GPR52 (0.67) GPR52S1PR4S1PR5ALDH1A1
SCHEMBL3209846 0.84 GPR52 (0.69) GPR52S1PR4S1PR5ALDH1A1
SCHEMBL1847987 0.83 GPR52 (0.48) GPR52S1PR4S1PR5ALDH1A1MEN1
SCHEMBL1847683 0.82 MAPT (0.50) GPR52ALDH1A1MEN1KMT2ARAB9A
SCHEMBL3206663 0.81 GPR52 (0.68) GPR52S1PR4S1PR5ALDH1A1
SCHEMBL3221889 0.79 GPR52 (0.71) GPR52S1PR4S1PR5ALDH1A1
SCHEMBL1850455 0.79 GPR52 (0.49) GPR52S1PR4S1PR5DHODHALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed