SCHEMBL1850455

SCHEMBL1850455

NC(=O)c1cccc(-c2cccc3cc(C(O)c4cccc(C(F)(F)F)c4)sc23)c1.O=C(O)c1cccc(-c2cccc3cc(C(O)c4cccc(C(F)(F)F)c4)sc23)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 4/20 0.49
DHODH Q02127 1/20 0.43
S1PR4 O95977 2/20 0.42
S1PR5 Q9H228 2/20 0.42
AKR1C3 P42330 3/20 0.39
AKR1C2 P52895 3/20 0.39
CES2 O00748 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
CFTR P13569 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SCD O00767 1/20 0.37
PLG P00747 1/20 0.37
PLAU P00749 1/20 0.37
PLAT P00750 1/20 0.37
SLC9A1 P19634 1/20 0.36
SRD5A2 P31213 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3219110 0.96 GPR52 (0.51) GPR52DHODHS1PR4S1PR5AKR1C3
SCHEMBL3198656 0.95 GPR52 (0.49) GPR52S1PR4S1PR5AKR1C3AKR1C2
SCHEMBL1850452 0.89 GPR52 (0.46) GPR52DHODHS1PR4S1PR5AKR1C3
SCHEMBL1849541 0.88 GPR52 (0.66) GPR52S1PR4S1PR5ALDH1A1SCD
SCHEMBL3206554 0.85 GPR52 (0.46) GPR52S1PR4S1PR5AKR1C3AKR1C2
SCHEMBL3198211 0.84 GPR52 (0.70) GPR52S1PR4S1PR5ALDH1A1SCD
SCHEMBL1850454 0.83 MAPT (0.52) GPR52MEN1KMT2AALDH1A1RAB9A
SCHEMBL3204669 0.83 GPR52 (0.49) GPR52S1PR4S1PR5CES2MEN1
SCHEMBL3209079 0.81 GPR52 (0.70) GPR52S1PR4S1PR5ALDH1A1SCD
SCHEMBL1849010 0.80 GPR52 (0.54) GPR52S1PR4S1PR5MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed