SCHEMBL1847713

SCHEMBL1847713

O=C(O)c1cccc(-c2cccc3cc(CCc4cccc(C(F)(F)F)c4)sc23)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 9/20 0.62
S1PR5 Q9H228 4/20 0.55
S1PR4 O95977 2/20 0.55
NR4A2 P43354 2/20 0.46
MRGPRX4 Q96LA9 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
KMT2A Q03164 1/20 0.43
LIPG Q9Y5X9 1/20 0.42
PTPRC P08575 1/20 0.41
PTPN2 P17706 1/20 0.41
PTPN1 P18031 1/20 0.41
PTPN6 P29350 1/20 0.41
PTPN9 P43378 1/20 0.41
DUSP3 P51452 1/20 0.41
PTPN11 Q06124 1/20 0.41
PTPN22 Q9Y2R2 1/20 0.41
S1PR1 P21453 1/20 0.41
GRK5 P34947 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1853402 0.91 GPR52 (0.75) GPR52S1PR5S1PR4NR4A2
SCHEMBL1850704 0.88 GPR52 (0.60) GPR52S1PR5S1PR4KDM4EMEN1
SCHEMBL1854351 0.85 GPR52 (0.85) GPR52S1PR5S1PR4MRGPRX4CDK8
SCHEMBL1849956 0.84 GPR52 (0.86) GPR52S1PR5S1PR4MRGPRX4
SCHEMBL1854277 0.82 S1PR5 (0.63) GPR52S1PR5S1PR4LIPG
SCHEMBL1849010 0.82 GPR52 (0.54) GPR52S1PR5S1PR4NR4A2MRGPRX4
SCHEMBL1850062 0.82 MRGPRX4 (0.57) GPR52S1PR5S1PR4NR4A2MRGPRX4
SCHEMBL1852578 0.82 GPR52 (0.61) GPR52S1PR5S1PR4
SCHEMBL1852567 0.82 GPR52 (0.78) GPR52S1PR5S1PR4
SCHEMBL1853172 0.81 GPR52 (0.67) GPR52S1PR5S1PR4NR4A2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed