SCHEMBL1849010

SCHEMBL1849010

O=C(O)c1cccc(-c2cccc3cc(C(O)Cc4cccc(C(F)(F)F)c4)sc23)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 7/20 0.54
S1PR4 O95977 2/20 0.48
S1PR5 Q9H228 2/20 0.48
NR4A2 P43354 2/20 0.44
MRGPRX4 Q96LA9 1/20 0.42
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
KMT2A Q03164 1/20 0.41
USP2 O75604 2/20 0.41
CYP3A4 P08684 2/20 0.41
NR1I2 O75469 1/20 0.41
ADRB1 P08588 1/20 0.41
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
CHRM3 P20309 1/20 0.41
SLC6A2 P23975 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3198656 0.84 GPR52 (0.49) GPR52S1PR4S1PR5KDM4EMEN1
SCHEMBL1853402 0.83 GPR52 (0.75) GPR52S1PR4S1PR5NR4A2
SCHEMBL1847713 0.82 GPR52 (0.62) GPR52S1PR4S1PR5NR4A2MRGPRX4
SCHEMBL1849012 0.82 GPR52 (0.53) GPR52S1PR4S1PR5KDM4EMEN1
SCHEMBL3206554 0.81 GPR52 (0.46) GPR52S1PR4S1PR5KDM4EMEN1
SCHEMBL1848384 0.80 GPR52 (0.65) GPR52S1PR4S1PR5MRGPRX4
SCHEMBL1850455 0.80 GPR52 (0.49) GPR52S1PR4S1PR5KDM4EMEN1
SCHEMBL1853719 0.77 GPR52 (0.44) GPR52S1PR4S1PR5KDM4EMEN1
SCHEMBL1852737 0.77 HTR2A (0.45) USP2CYP3A4NR1I2ADRB1HTR1A
SCHEMBL1849541 0.77 GPR52 (0.66) GPR52S1PR4S1PR5MRGPRX4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed