SCHEMBL18487394

SCHEMBL18487394

Cc1cc(F)cc(-c2nccc(N)c2N)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.36
ADORA1 P30542 5/20 0.36
TDO2 P48775 2/20 0.36
NOS3 P29474 2/20 0.35
NOS2 P35228 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
NOS1 P29475 1/20 0.35
KMT2A Q03164 1/20 0.35
BACE1 P56817 2/20 0.34
PDE10A Q9Y233 1/20 0.34
LRRK2 Q5S007 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28704506 0.81 ADORA2A (0.39) ADORA2AADORA1TDO2BACE1PDE10A
SCHEMBL17555820 0.81 KDM1A (0.42) TDO2BACE1
SCHEMBL17555811 0.80 KDM1A (0.45) ADORA2AADORA1NOS3NOS2NOS1
SCHEMBL17555819 0.77 TDO2 (0.48) ADORA2AADORA1TDO2KDM4EMEN1
SCHEMBL17555834 0.75 PDE3B (0.42) ADORA2AADORA1
SCHEMBL18474589 0.74 NOS3 (0.43) NOS3NOS2KDM4EMEN1NOS1
SCHEMBL16805988 0.74 PDE10A (0.37) ADORA2AADORA1PDE10ALRRK2ADORA3
SCHEMBL17555926 0.74 ADORA2A (0.41) ADORA2AADORA1
SCHEMBL18486943 0.73 NOS1 (0.46) NOS3NOS2NOS1
SCHEMBL17568762 0.73 MAP4K4 (0.48) TDO2NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017023972-A1 3-(1H-IMIDAZO[4,5-C]PYRIDIN-2-YL)-1H-PYRAZOLO[4,3-B]PYRIDINES AND THERAPEUTIC USES THEREOF SAMUMED, LLC. (US) 2017-02-09 WO disclosed