SCHEMBL18487537

SCHEMBL18487537

COc1ccc2c(c1)[nH]c1ccc(OSc3cccc4c(N(C)C)cccc34)cc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
KDM4E B2RXH2 2/20 0.50
MEN1 O00255 2/20 0.50
MAPT P10636 2/20 0.50
KMT2A Q03164 2/20 0.50
HSD17B10 Q99714 2/20 0.50
HPGD P15428 1/20 0.50
TSHR P16473 1/20 0.46
GFER P55789 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.41
CHUK O15111 1/20 0.40
ACHE P22303 3/20 0.39
BCHE P06276 1/20 0.39
HTR7 P34969 3/20 0.36
HTR1A P08908 2/20 0.36
HTR1D P28221 2/20 0.36
HTR5A P47898 2/20 0.36
HTR6 P50406 2/20 0.36
SLC6A4 P31645 1/20 0.36
GABRP O00591 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18487745 0.84 DYRK1A (0.40) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL18487739 0.81 DYRK1A (0.40) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL18487536 0.77 KDM4E (0.48) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL1181326 0.69 KDM4E (0.79) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL29670412 0.69 KDM4E (0.79) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL532262 0.69 ALDH1A1 (1.00) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL29562964 0.69 ALDH1A1 (1.00) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL30115280 0.69 KDM4E (0.79) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL29643258 0.69 ALDH1A1 (1.00) ALDH1A1KDM4EMEN1MAPTKMT2A
7-Methoxy-3-Methylcarbazole SCHEMBL31214611 0.68 KDM4E (0.67) ALDH1A1KDM4EMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017023916-A1 SMALL MOLECULE ANDROGEN RECEPTOR INHIBITORS AND METHODS OF USE THEREOF GEORGETOWN UNIVERSITY (US) 2017-02-09 WO disclosed