SCHEMBL18488024

SCHEMBL18488024

NC(c1cc(Br)ccc1F)C(F)F

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.37
DGAT1 O75907 1/20 0.36
KDM1A O60341 2/20 0.34
KDM1B Q8NB78 1/20 0.34
APLNR P35414 2/20 0.33
ALOX5AP P20292 1/20 0.30
FEN1 P39748 1/20 0.30
IDO1 P14902 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18449718 1.00 DPP4 (0.37) DPP4DGAT1KDM1AKDM1BAPLNR
SCHEMBL18449939 1.00 DPP4 (0.37) DPP4DGAT1KDM1AKDM1BAPLNR
SCHEMBL20256754 0.81 DPP4 (0.40) DPP4DGAT1KDM1AKDM1BAPLNR
SCHEMBL248835 0.81 DGAT1 (0.38) DPP4DGAT1KDM1AKDM1BAPLNR
SCHEMBL29604357 0.81 DGAT1 (0.38) DPP4DGAT1KDM1AKDM1BAPLNR
SCHEMBL29668972 0.79 CES2 (0.42) DPP4KDM1AKDM1BIDO1
SCHEMBL20238308 0.79 CES2 (0.42) DPP4KDM1AKDM1BIDO1
SCHEMBL20238309 0.79 CES2 (0.42) DPP4KDM1AKDM1BIDO1
SCHEMBL14987514 0.78 PDE2A (0.43) DPP4DGAT1KDM1AKDM1BAPLNR
SCHEMBL20238210 0.78 PDE2A (0.43) DPP4DGAT1KDM1AKDM1BAPLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137547-B Heterocyclic compounds useful as TNF alpha modulators 百时美施贵宝公司 2021-11-12 CN disclosed
WO-2017023905-A1 HETEROCYCLIC COMPOUNDS USEFUL AS MODULATORS OF TNF ALPHA BRISTOL-MYERS SQUIBB COMPANY (US) 2017-02-09 WO disclosed