SCHEMBL1850163

SCHEMBL1850163

CCOC(=O)c1cccc(-c2cccc3nn(Cc4cc(F)cc(Cl)c4)cc23)c1.Fc1cc(Cl)cc(Cn2cc3c(Br)cccc3n2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 2/20 0.45
JMJD6 Q6NYC1 2/20 0.38
KLKB1 P03952 1/20 0.37
TP53 P04637 1/20 0.37
GRM2 Q14416 1/20 0.36
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
PRKDC P78527 1/20 0.35
AGTR1 P30556 1/20 0.35
CYP19A1 P11511 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
UBE2N P61088 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1853574 0.95 GPR52 (0.48) GPR52JMJD6KLKB1TP53GRM2
SCHEMBL1849622 0.90 GPR52 (0.51) GPR52JMJD6KLKB1TP53GRM2
SCHEMBL1857340 0.89 GPR52 (0.46) GPR52JMJD6KLKB1TP53GRM2
SCHEMBL1849364 0.86 GPR52 (0.51) GPR52JMJD6GRM2ALDH1A1SMN1; SMN2
SCHEMBL3215484 0.85 GPR52 (0.55) GPR52JMJD6KLKB1TP53GRM2
SCHEMBL1852588 0.85 GPR52 (0.53) GPR52JMJD6KLKB1TP53ALDH1A1
SCHEMBL3217768 0.83 GPR52 (0.50) GPR52JMJD6KLKB1TP53GRM2
SCHEMBL1848441 0.83 GPR52 (0.50) GPR52SMN1; SMN2NPC1RAB9A
SCHEMBL1856096 0.83 GPR52 (0.54) GPR52JMJD6ALDH1A1MAPTSMN1; SMN2
SCHEMBL1851052 0.82 GPR52 (0.58) GPR52KLKB1MAPTSMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed