SCHEMBL1851052

SCHEMBL1851052

O=C(NCCOC(=O)c1cccc(-c2cccc3nn(Cc4cc(F)cc(Cl)c4)cc23)c1)c1cccc(-c2cccc3nn(Cc4cc(F)cc(Cl)c4)cc23)c1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 5/20 0.58
KLKB1 P03952 6/20 0.40
DGAT2 Q96PD7 1/20 0.38
ADORA3 P0DMS8 1/20 0.37
ADORA2B P29275 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
KMT2A Q03164 2/20 0.37
AURKA O14965 1/20 0.36
KDM4E B2RXH2 2/20 0.36
MAPT P10636 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1852544 0.91 GPR52 (0.62) GPR52KLKB1DGAT2ADORA3ADORA2B
SCHEMBL1853932 0.90 GPR52 (0.63) GPR52KLKB1ADORA3ADORA2BSMN1; SMN2
SCHEMBL3209129 0.89 GPR52 (0.69) GPR52ADORA3ADORA2BAURKA
SCHEMBL1853574 0.87 GPR52 (0.48) GPR52KLKB1SMN1; SMN2MAPT
SCHEMBL1851055 0.86 GPR52 (0.65) GPR52ADORA3ADORA2B
SCHEMBL3208468 0.86 GPR52 (0.57) GPR52KLKB1ADORA3ADORA2BAURKA
SCHEMBL1849604 0.84 GPR52 (0.81) GPR52ADORA3CYP1A2CYP3A4CYP2D6
SCHEMBL1848441 0.83 GPR52 (0.50) GPR52ADORA3ADORA2BSMN1; SMN2CYP2C9
SCHEMBL1850163 0.82 GPR52 (0.45) GPR52KLKB1SMN1; SMN2KMT2AKDM4E
SCHEMBL1850671 0.82 GPR52 (0.62) GPR52KLKB1DGAT2KMT2AAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed