SCHEMBL1850479

SCHEMBL1850479

CS(=O)(=O)c1cccc(Cc2cc3c(F)ccc(-c4cccc(C(=O)O)c4)c3s2)c1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 6/20 0.53
PLA2G2A P14555 1/20 0.41
PTGER1 P34995 5/20 0.41
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
PARP1 P09874 1/20 0.37
CAMKK2 Q96RR4 1/20 0.37
FOLH1 Q04609 1/20 0.36
KAT6A Q92794 1/20 0.35
CSNK2A2 P19784 1/20 0.35
CSNK2B P67870 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1851664 0.88 GPR52 (0.51) GPR52ALDH1A1CA2
SCHEMBL1852822 0.86 GPR52 (0.73) GPR52ALDH1A1GAAHSD17B10PARP1
SCHEMBL1848566 0.85 GPR52 (0.59) GPR52ALDH1A1GAAHSD17B10
SCHEMBL3213715 0.85 GPR52 (0.56) GPR52PLA2G2APTGER1AKR1C3AKR1C2
SCHEMBL1848214 0.82 GPR52 (0.74) GPR52PLA2G2AAKR1C3AKR1C2ALDH1A1
SCHEMBL1849783 0.79 GPR52 (0.56) GPR52PLA2G2APTGER1AKR1C3AKR1C2
SCHEMBL1850572 0.79 GPR52 (0.74) GPR52PLA2G2A
SCHEMBL1847069 0.78 GPR52 (0.36) GPR52ALDH1A1GAAHSD17B10PARP1
SCHEMBL1848607 0.78 GPR52 (0.56) GPR52PTGER1
SCHEMBL3208322 0.77 GPR52 (0.49) GPR52PLA2G2APTGER1AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed