SCHEMBL1850671

SCHEMBL1850671

COc1cccc(Cn2cc3c(-c4cccc(C(=O)NCCOC(=O)c5cccc(-c6cccc7nn(Cc8cccc(OC)c8)cc67)c5)c4)cccc3n2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 2/20 0.62
MMP13 P45452 2/20 0.45
DGAT2 Q96PD7 1/20 0.45
KLKB1 P03952 1/20 0.45
AURKA O14965 1/20 0.44
PTGER4 P35408 1/20 0.43
SMYD2 Q9NRG4 1/20 0.43
KMT2A Q03164 1/20 0.42
TP53 P04637 2/20 0.42
ALDH1A1 P00352 1/20 0.41
PTAFR P25105 1/20 0.41
CHRM3 P20309 1/20 0.41
CDC7 O00311 1/20 0.40
DAPK3 O43293 1/20 0.40
JAK2 O60674 1/20 0.40
ROCK2 O75116 1/20 0.40
MAP4K4 O95819 1/20 0.40
PAK4 O96013 1/20 0.40
PRKACA P17612 1/20 0.40
CDK2 P24941 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3219552 0.90 GPR52 (0.73) GPR52MMP13DGAT2AURKAPTGER4
SCHEMBL1853932 0.88 GPR52 (0.63) GPR52KLKB1PTGER4KMT2ATP53
SCHEMBL1850607 0.87 GPR52 (0.52) GPR52KLKB1PTGER4KMT2ATP53
SCHEMBL1849604 0.87 GPR52 (0.81) GPR52PTGER4ALDH1A1CHRM3
SCHEMBL1850675 0.87 GPR52 (0.69) GPR52MMP13DGAT2AURKAPTGER4
SCHEMBL3217756 0.87 GPR52 (0.59) GPR52MMP13DGAT2AURKAPTGER4
SCHEMBL1852544 0.86 GPR52 (0.62) GPR52DGAT2KLKB1PTGER4KMT2A
SCHEMBL1848805 0.85 GPR52 (0.53) GPR52KLKB1KMT2AROCK2
SCHEMBL1857499 0.84 GPR52 (0.56) GPR52MMP13DGAT2AURKAPTGER4
SCHEMBL1853272 0.83 GPR52 (0.53) GPR52MMP13DGAT2PTGER4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed