SCHEMBL1849604

SCHEMBL1849604

O=C(NCCOC(=O)c1cccc(-c2cccc3nn(Cc4cccc(C(F)(F)F)c4)cc23)c1)c1cccc(-c2cccc3nn(Cc4cccc(C(F)(F)F)c4)cc23)c1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 13/20 0.81
PTGER4 P35408 1/20 0.43
USP2 O75604 2/20 0.41
CYP3A4 P08684 2/20 0.41
CHRM3 P20309 2/20 0.41
NR1I2 O75469 1/20 0.41
ADRB1 P08588 1/20 0.41
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
SLC6A2 P23975 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
SLC6A4 P31645 1/20 0.41
ADRA1A P35348 1/20 0.41
HRH1 P35367 1/20 0.41
OPRM1 P35372 1/20 0.41
DRD3 P35462 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3207056 0.90 GPR52 (1.00) GPR52PTGER4CHRM3ALDH1A1POLB
SCHEMBL1853932 0.88 GPR52 (0.63) GPR52PTGER4ADORA3
SCHEMBL1852544 0.87 GPR52 (0.62) GPR52PTGER4CYP3A4ADORA3CYP1A2
SCHEMBL1851622 0.87 GPR52 (0.81) GPR52USP2CYP3A4CHRM3NR1I2
SCHEMBL1849610 0.87 GPR52 (0.93) GPR52PTGER4
SCHEMBL1850671 0.87 GPR52 (0.62) GPR52PTGER4CHRM3ALDH1A1
SCHEMBL3206470 0.87 GPR52 (0.81) GPR52PTGER4CHRM3ALDH1A1POLB
SCHEMBL1851194 0.86 GPR52 (0.70) GPR52PTGER4ALDH1A1
SCHEMBL1856279 0.84 GPR52 (0.77) GPR52PTGER4
SCHEMBL1851052 0.84 GPR52 (0.58) GPR52CYP3A4ADORA3CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed