SCHEMBL1852544

SCHEMBL1852544

O=C(NCCOC(=O)c1cccc(-c2cccc3nn(Cc4ccc(F)cc4)cc23)c1)c1cccc(-c2cccc3nn(Cc4ccc(F)cc4)cc23)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 4/20 0.62
KMT2A Q03164 1/20 0.43
DGAT2 Q96PD7 1/20 0.42
MAPT P10636 2/20 0.42
KDM4E B2RXH2 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
KLKB1 P03952 4/20 0.40
PTGER4 P35408 3/20 0.40
ADORA3 P0DMS8 1/20 0.38
ADORA2B P29275 1/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 1/20 0.38
TP53 P04637 1/20 0.37
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1851052 0.91 GPR52 (0.58) GPR52KMT2ADGAT2MAPTKDM4E
SCHEMBL1853932 0.89 GPR52 (0.63) GPR52KMT2AMAPTKDM4EKLKB1
SCHEMBL3217594 0.88 GPR52 (0.75) GPR52PTGER4ADORA3ADORA2B
SCHEMBL1849604 0.87 GPR52 (0.81) GPR52CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL1850671 0.86 GPR52 (0.62) GPR52KMT2ADGAT2KLKB1PTGER4
SCHEMBL1849364 0.86 GPR52 (0.51) GPR52ALDH1A1
SCHEMBL1850719 0.85 GPR52 (0.61) GPR52DGAT2MAPTPTGER4ADORA3
SCHEMBL1852548 0.85 GPR52 (0.70) GPR52PTGER4ADORA3ADORA2B
SCHEMBL1848805 0.82 GPR52 (0.53) GPR52KMT2AMAPTKDM4EKLKB1
SCHEMBL1850248 0.81 GPR52 (0.54) GPR52PTGER4ADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed