SCHEMBL18508246

SCHEMBL18508246

CNc1ccc(Br)cc1N[C@@H](C)COC

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.41
ALDH1A1 P00352 5/20 0.41
HCAR3 P49019 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
CYP2D6 P10635 1/20 0.33
HPGD P15428 3/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
POLB P06746 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
RECQL P46063 1/20 0.32
BLM P54132 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
LPAR1 Q92633 1/20 0.31
HSD17B10 Q99714 1/20 0.31
LMNA P02545 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18508300 1.00 KDM4E (0.41) KDM4EALDH1A1HCAR3TDP1CYP2D6
SCHEMBL18496294 0.81 ALDH1A1 (0.41) KDM4EALDH1A1HCAR3TDP1CYP2D6
SCHEMBL18496296 0.81 ALDH1A1 (0.41) KDM4EALDH1A1HCAR3TDP1CYP2D6
SCHEMBL29719399 0.81 ALDH1A1 (0.41) KDM4EALDH1A1HCAR3TDP1CYP2D6
SCHEMBL18508189 0.81 ALDH1A1 (0.41) KDM4EALDH1A1HCAR3TDP1CYP2D6
SCHEMBL4580624 0.78 KDM4E (0.39) KDM4EALDH1A1HCAR3TDP1HPGD
SCHEMBL29719195 0.76 HCAR3 (0.57) KDM4EALDH1A1HCAR3TDP1CYP2D6
SCHEMBL18496291 0.76 HCAR3 (0.57) KDM4EALDH1A1HCAR3TDP1CYP2D6
SCHEMBL18496278 0.76 HCAR3 (0.57) KDM4EALDH1A1HCAR3TDP1CYP2D6
SCHEMBL18496289 0.76 HCAR3 (0.57) KDM4EALDH1A1HCAR3TDP1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017024412-A1 SUBSTITUTED BENZIMIDAZOLES, THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS NEOMED INSTITUTE (CA) 2017-02-16 WO disclosed