SCHEMBL1850828

SCHEMBL1850828

COc1cccc(Cc2cc3cccc(-c4cccc(C(=O)N(CCN5CCCC5)c5cccc(-c6cccc7cc(Cc8cccc(OC)c8)oc67)c5)c4)c3o2)c1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.44
ALDH1A1 P00352 2/20 0.42
SMYD2 Q9NRG4 1/20 0.42
HPGD P15428 1/20 0.42
KDM4E B2RXH2 1/20 0.41
GPR52 Q9Y2T5 1/20 0.41
ROCK2 O75116 5/20 0.39
ROCK1 Q13464 5/20 0.39
HTR2B P41595 2/20 0.39
ADRA2A P08913 1/20 0.39
HTR2A P28223 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
DRD4 P21917 1/20 0.39
LTA4H P09960 1/20 0.38
PTGIR P43119 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
WDR5 P61964 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3211200 0.83 SMYD2 (0.57) SMYD2GPR52DRD4
SCHEMBL1850827 0.80 SMYD2 (0.54) SMYD2GPR52DRD4
SCHEMBL1849693 0.78 GPR52 (0.52) GPR52
SCHEMBL1855790 0.74 GPR52 (0.45) ALDH1A1HPGDGPR52
SCHEMBL1851120 0.73 GPR52 (0.53) ALDH1A1SMYD2GPR52DRD4
SCHEMBL1849845 0.72 GPR52 (0.44) ALDH1A1HPGDKDM4EGPR52
SCHEMBL1855327 0.71 GPR52 (0.51) ALDH1A1GPR52DRD4
SCHEMBL7959088 0.70 TAS1R3 (0.53) HPGDGPR52
SCHEMBL1850921 0.68 GPR52 (0.49) ALDH1A1HPGDGPR52ROCK2ROCK1
SCHEMBL3209922 0.67 GPR52 (0.49) HPGDKDM4EGPR52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed