SCHEMBL18516616

SCHEMBL18516616

Cc1cccc(CN(C)CCN2CCN(C)CC2)c1

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 13/20 0.62
HRH3 Q9Y5N1 1/20 0.53
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
RECQL P46063 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.45
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10288974 0.85 SIGMAR1 (0.62) SIGMAR1KDM4EALDH1A1
SCHEMBL18516696 0.83 SIGMAR1 (0.60) SIGMAR1HRH3ALDH1A1
SCHEMBL10223554 0.81 SIGMAR1 (0.58) SIGMAR1
SCHEMBL18516615 0.81 SIGMAR1 (0.58) SIGMAR1ALDH1A1
SCHEMBL18516703 0.81 SIGMAR1 (0.58) SIGMAR1
SCHEMBL12880000 0.81 HRH3 (0.78) SIGMAR1HRH3CYP2D6L3MBTL1KDM4E
SCHEMBL10076573 0.79 MC4R (0.65) HRH3CYP2D6CYP2C19KDM4EALDH1A1
SCHEMBL18378603 0.77 CYP2D6 (0.57) SIGMAR1CYP2D6CYP2C9CYP2C19RECQL
SCHEMBL18138028 0.77 CYP2D6 (0.57) SIGMAR1CYP2D6CYP2C9CYP2C19RECQL
SCHEMBL13675505 0.77 SIGMAR1 (0.71) SIGMAR1CYP2D6KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957498-B1 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING METHYLGENE INC (CA) 2017-02-15 EP disclosed