SCHEMBL18518271

SCHEMBL18518271

CN1CCCC(Nc2ncnc(N)c2C(=N)c2cc(-c3ccccc3)on2)C1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 2/20 0.44
LRRK2 Q5S007 1/20 0.42
BTK Q06187 3/20 0.41
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
KAT2B Q92831 2/20 0.40
S1PR1 P21453 1/20 0.40
EGFR P00533 1/20 0.39
NLRP3 Q96P20 1/20 0.38
SCD5 Q86SK9 5/20 0.38
SCD O00767 1/20 0.38
USP30 Q70CQ3 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18518275 0.83 CSF1R (0.48) BTKNPC1RAB9ASMN1; SMN2S1PR1
SCHEMBL19649120 0.78 BTK (0.61) BTKKAT2BEGFR
SCHEMBL24196488 0.78 BTK (0.61) BTKKAT2BEGFR
SCHEMBL21899550 0.76 BTK (0.44) CHEK1LRRK2BTKKAT2BEGFR
SCHEMBL18518831 0.76 ALDH1A1 (0.50) NPC1RAB9ASMN1; SMN2S1PR1SCD5
SCHEMBL25060362 0.72 BTK (0.59) CHEK1LRRK2BTKKAT2BEGFR
SCHEMBL18518280 0.71 NPC1 (0.39) NPC1RAB9ASMN1; SMN2S1PR1HPGD
SCHEMBL22243292 0.69 BTK (0.45) BTKNPC1RAB9ASMN1; SMN2EGFR
SCHEMBL24380910 0.69 BTK (0.61) BTKEGFR
SCHEMBL23223035 0.68 BTK (0.46) CHEK1LRRK2BTKKAT2BEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017026718-A1 NOVEL 3-(ISOXAZOL-3-YL)-PYRAZOLO[3,4-D]PYRIMIDIN-4-AMINE COMPOUND, WHICH IS RET KINASE INHIBITOR 한국과학기술연구원 2017-02-16 WO disclosed