SCHEMBL21899550

SCHEMBL21899550

CN1CCCC(Nc2ncnc(N)c2C(=N)Br)C1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BTK Q06187 3/20 0.44
KAT2B Q92831 5/20 0.43
LRRK2 Q5S007 1/20 0.41
NLRP3 Q96P20 1/20 0.38
CHEK1 O14757 1/20 0.38
JAK3 P52333 5/20 0.37
IL1B P01584 4/20 0.37
BPTF Q12830 1/20 0.37
EGFR P00533 1/20 0.37
JAK1 P23458 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21899804 0.84 BTK (0.47) BTKJAK3EGFRJAK1
SCHEMBL24464321 0.82 HPGDS (0.44) EGFRJAK1
SCHEMBL14647420 0.80 BTK (0.50) BTKJAK3EGFRJAK1
SCHEMBL21900351 0.79 BTK (0.49) BTKJAK3EGFRJAK1
SCHEMBL21899548 0.78 BTK (0.49) BTKJAK3EGFRJAK1
SCHEMBL21159574 0.78 KAT2B (0.46) BTKKAT2BLRRK2NLRP3CHEK1
SCHEMBL24196488 0.78 BTK (0.61) BTKKAT2BEGFR
SCHEMBL19649120 0.78 BTK (0.61) BTKKAT2BEGFR
SCHEMBL26411460 0.76 PIK3CD (0.42) BTKKAT2B
SCHEMBL18518271 0.76 CHEK1 (0.44) BTKKAT2BLRRK2NLRP3CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3257855-B1 METHOD FOR PREPARING IBRUTINIB SHANGHAI DUDE MEDICAL SCIENCE AND TECH CO LTD (CN) 2020-04-22 EP disclosed