SCHEMBL18525995

SCHEMBL18525995

Cc1cc(CN(C)F)cc(C(C)C)n1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
GSR P00390 1/20 0.33
TSHR P16473 3/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TLR9 Q9NR96 1/20 0.31
TLR8 Q9NR97 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
ALDH1A1 P00352 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CRHBP P24387 1/20 0.30
CYP2C19 P33261 1/20 0.30
CRHR2 Q13324 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18525716 0.76 NOS3 (0.39) NOS3NOS1NOS2TSHRMAPT
SCHEMBL18489378 0.74 NOS3 (0.42) NOS3NOS1NOS2TSHRKMT2A
SCHEMBL18489341 0.74 NOS3 (0.38) NOS3NOS1NOS2TSHRKMT2A
SCHEMBL23280272 0.71 NOS3 (0.36) NOS3NOS1NOS2TSHRMAPT
SCHEMBL15980633 0.68 NOS3 (0.39) NOS3NOS1NOS2TSHRKMT2A
SCHEMBL20063092 0.67 NOS3 (0.42) NOS3NOS1NOS2TSHRKMT2A
SCHEMBL23287928 0.66 ALDH1A1 (0.42) NOS3NOS1NOS2GSRTSHR
SCHEMBL4547885 0.66 NOS2 (0.61) NOS3NOS1NOS2TSHRKMT2A
SCHEMBL18792891 0.66 HMGCR (0.35) NOS3NOS1NOS2
SCHEMBL20356746 0.66 KDM5A (0.33) NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017027343-A1 CGRP RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2017-02-16 WO disclosed