SCHEMBL18535017

SCHEMBL18535017

CNc1cc(C#N)ccc1C(=N)c1cnc2c(n1)c(C(=O)NC(C)(C)C)cn2COC(=O)C(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 6/20 0.35
LRRK2 Q5S007 1/20 0.32
ANO1 Q5XXA6 1/20 0.32
TNF P01375 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18535076 0.94 SCN9A (0.36) IRAK4
SCHEMBL18534974 0.83 NR3C1 (0.30)
SCHEMBL18535004 0.80 MAPT (0.31)
SCHEMBL18535027 0.79 ALDH1A1 (0.31)
SCHEMBL18535276 0.78 CFTR (0.34)
SCHEMBL18535101 0.78 KDM4E (0.40)
SCHEMBL18535117 0.77 SYK (0.49)
SCHEMBL14737367 0.76 SYK (0.48)
SCHEMBL14751406 0.73 TLR2 (0.36)
SCHEMBL14738395 0.73 ABCB11 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2763990-B1 PYRROLOPYRAZINE KINASE INHIBITORS HOFFMANN LA ROCHE (CH) 2017-02-22 EP disclosed