SCHEMBL18540697

SCHEMBL18540697

N=C(c1cccc(O)c1)c1cccc(Br)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
C1S P09871 1/20 0.57
CTSL P07711 3/20 0.50
PARP1 P09874 2/20 0.47
KDM4E B2RXH2 2/20 0.46
EGLN2 Q96KS0 1/20 0.46
CA12 O43570 2/20 0.45
CA2 P00918 2/20 0.45
CA9 Q16790 2/20 0.45
CA1 P00915 1/20 0.45
CA6 P23280 1/20 0.45
MAPT P10636 2/20 0.43
AKR1C4 P17516 1/20 0.43
AKR1C3 P42330 1/20 0.43
AKR1C2 P52895 1/20 0.43
AKR1C1 Q04828 1/20 0.43
MEN1 O00255 1/20 0.43
ABL1 P00519 1/20 0.43
TSHR P16473 1/20 0.43
KMT2A Q03164 1/20 0.43
RIN1 Q13671 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18540679 0.90 C1S (0.55) C1SCTSLPARP1MAPTMEN1
SCHEMBL30136033 0.80 FASN (0.61) CTSLPARP1KDM4EEGLN2CA12
SCHEMBL4511367 0.80 PARP1 (0.57) C1SCTSLPARP1KDM4EEGLN2
SCHEMBL18529814 0.80 FASN (0.61) CTSLPARP1KDM4EEGLN2CA12
SCHEMBL29505543 0.78
SCHEMBL49927 0.78
SCHEMBL931503 0.77 C1S (0.53) C1SCTSLPARP1MEN1KMT2A
SCHEMBL932511 0.77 C1S (0.53) C1SCTSLPARP1MAPTMEN1
SCHEMBL31174803 0.76 CTSL (0.61) C1SCTSLPARP1KDM4EEGLN2
Phosphine SCHEMBL4337915 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017030983-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF CATHEPSINS MATEON THERAPEUTICS, INC. (US) 2017-02-23 WO disclosed