SCHEMBL18544282

SCHEMBL18544282

COc1ccc2c(F)ccc(I)c2n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
KMT2A Q03164 1/20 0.38
MAPK13 O15264 1/20 0.36
MAPK12 P53778 1/20 0.36
MAPK11 Q15759 1/20 0.36
MAPK14 Q16539 1/20 0.36
DYRK1A Q13627 4/20 0.36
CLK1 P49759 2/20 0.36
CLK2 P49760 1/20 0.36
CLK3 P49761 1/20 0.36
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
MTNR1A P48039 2/20 0.35
MTNR1B P49286 2/20 0.35
TDO2 P48775 1/20 0.33
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA2 P47869 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25097019 0.79 CYP1A2 (0.38) CYP1A2KMT2ADYRK1ACLK1CLK2
SCHEMBL20687488 0.78 KMT2A (0.35) CYP1A2KMT2AMAPK13MAPK12MAPK11
SCHEMBL18544258 0.77 CYP1A2 (0.40) CYP1A2KMT2AMAPK13MAPK12MAPK11
SCHEMBL2461286 0.75 POLB (0.36) CYP1A2KMT2AMAPK13MAPK12MAPK11
Hydrochloric Acid SCHEMBL20563346 0.74 MTNR1A (0.38) KMT2AMTNR1AMTNR1B
SCHEMBL18544287 0.74 PTGS2 (0.37) CYP1A2KMT2AMTNR1AMTNR1BPOLB
SCHEMBL2172807 0.74 KMT2A (0.37) CYP1A2KMT2AMAPK13MAPK12MAPK11
SCHEMBL18544275 0.74 CYP11B2 (0.33)
SCHEMBL17543401 0.74 CYP1A2 (0.37) CYP1A2KMT2AMAPK13MAPK12MAPK11
SCHEMBL2819275 0.70 PTGS2 (0.37) CYP1A2KMT2AMTNR1AMTNR1BPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017029602-A2 COMPOUNDS FOR USE IN ANTIBACTERIAL APPLICATIONS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-02-23 WO disclosed