SCHEMBL18550982

SCHEMBL18550982

CC(=O)OC1C=C(C#CS(C)(C)C)CC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.34
CA12 O43570 4/20 0.31
CA9 Q16790 4/20 0.31
LMNA P02545 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
MAPK1 P28482 1/20 0.31
CYP2C19 P33261 1/20 0.31
ABCB11 O95342 1/20 0.31
ESR1 P03372 1/20 0.31
PGR P06401 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
AR P10275 1/20 0.31
CHRM1 P11229 1/20 0.31
MAOA P21397 1/20 0.31
SLC6A2 P23975 1/20 0.31
PDE4A P27815 1/20 0.31
ADRA1A P35348 1/20 0.31
CA1 P00915 2/20 0.30
CA2 P00918 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21916428 1.00 CYP19A1 (0.34) CYP19A1CA12CA9LMNACYP3A4
SCHEMBL18550781 0.79 DRD2 (0.36) CYP19A1LMNACYP3A4CYP2C9MAPK1
SCHEMBL21833718 0.79 DRD2 (0.36) CYP19A1LMNACYP3A4CYP2C9MAPK1
SCHEMBL21833716 0.79 DRD2 (0.36) CYP19A1LMNACYP3A4CYP2C9MAPK1
SCHEMBL2585385 0.71 CYP19A1 (0.40) CYP19A1CA12CA9LMNACYP3A4
SCHEMBL13677475 0.71 CYP19A1 (0.40) CYP19A1LMNACYP3A4CYP2C9MAPK1
SCHEMBL4266335 0.71 CYP19A1 (0.40) CYP19A1CA12CA9LMNACYP3A4
SCHEMBL21916584 0.70
SCHEMBL23273202 0.67 OAT (0.42) CYP19A1LMNACYP3A4CYP2C9MAPK1
SCHEMBL399295 0.66 CYP19A1 (0.37) CYP19A1CA12CA9LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017029601-A1 HETEROARYL DERIVATIVES AS PARP INHIBITORS LUPIN LIMITED (IN) 2017-02-23 WO disclosed