SCHEMBL185517

SCHEMBL185517

COc1ncc(OC(=O)N[C@@]2(C(=O)NCc3ccc(Nc4ccc(F)cc4C(F)(F)F)cc3)CCOC2)cn1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 3/20 0.37
BTK Q06187 1/20 0.36
CNR2 P34972 3/20 0.34
KIT P10721 1/20 0.33
BDKRB1 P46663 1/20 0.33
PTGES O14684 1/20 0.33
FAAH O00519 2/20 0.33
PTK2 Q05397 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MAPK10 P53779 1/20 0.32
IDH1 O75874 1/20 0.32
TRPV1 Q8NER1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL185744 0.93 OPRL1 (0.36) OPRL1BTKCNR2BDKRB1FAAH
SCHEMBL185483 0.93 OPRL1 (0.38) OPRL1BTKCNR2BDKRB1FAAH
SCHEMBL186586 0.92 CNR2 (0.36) BTKCNR2BDKRB1PTGESPTK2
SCHEMBL186275 0.91 BTK (0.38) OPRL1BTKCNR2BDKRB1FAAH
SCHEMBL14856809 0.91 OPRL1 (0.35) OPRL1CNR2BDKRB1FAAHMAPK10
SCHEMBL199266 0.91 OPRL1 (0.36) OPRL1BTKCNR2BDKRB1PTGES
SCHEMBL186660 0.90 CNR2 (0.36) BTKCNR2BDKRB1FAAHPTK2
SCHEMBL186511 0.90 OPRL1 (0.39) OPRL1BTKCNR2FAAHPTK2
SCHEMBL2809806 0.90 BDKRB1 (0.38) OPRL1BTKCNR2KITBDKRB1
SCHEMBL185881 0.90 OPRL1 (0.37) OPRL1BTKCNR2BDKRB1FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-01-04 EP disclosed
WO-2010097372-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed