SCHEMBL18554238

SCHEMBL18554238

O=C(Nc1ccccc1C(=O)O)c1ncc[nH]1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.62
KMT2A Q03164 5/20 0.51
MEN1 O00255 4/20 0.51
PKM P14618 1/20 0.51
NPC1 O15118 3/20 0.51
ALDH1A1 P00352 3/20 0.51
RAB9A P51151 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
HPGD P15428 2/20 0.51
TP53 P04637 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C9 P11712 1/20 0.51
DHODH Q02127 1/20 0.50
CA12 O43570 1/20 0.49
CA2 P00918 1/20 0.49
CA9 Q16790 1/20 0.49
POLB P06746 1/20 0.46
KDM4D Q6B0I6 1/20 0.44
KDM4C Q9H3R0 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2817711 0.81 RAB9A (0.55) KMT2AMEN1PKMNPC1RAB9A
SCHEMBL13506700 0.81 HPGD (0.53) KMT2AMEN1PKMNPC1ALDH1A1
SCHEMBL7444006 0.80 RAB9A (0.50) KMT2AMEN1PKMNPC1ALDH1A1
SCHEMBL6906056 0.78 MAPT (0.49) KMT2AALDH1A1HPGDTP53CYP1A2
SCHEMBL12674223 0.77 MAPT (0.53) KMT2AALDH1A1CA12CA2CA9
SCHEMBL15165520 0.77 KDM4E (0.47) KMT2AALDH1A1
SCHEMBL9634432 0.77 ADRA2A (0.57) KMT2AMEN1ALDH1A1HPGDCYP1A2
SCHEMBL9542710 0.77 MAPT (0.48) KMT2AALDH1A1TP53CYP1A2CYP2C9
SCHEMBL2450877 0.76 KMT2A (0.69) NPSR1KMT2ANPC1ALDH1A1RAB9A
SCHEMBL2472433 0.76 MAPT (0.62) ALDH1A1SMN1; SMN2TP53CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3337795-A1 PIPERIDINOBENZODIAZEPINE COMPOUNDS WITH ANTI PROLIFERATIVE ACTIVITY Femtogenix Limited (GB) 2018-06-27 EP disclosed
WO-2017032983-A1 PIPERIDINOBENZODIAZEPINE COMPOUNDS WITH ANTI PROLIFERATIVE ACTIVITY FEMTOGENIX LIMITED (GB) 2017-03-02 WO disclosed