SCHEMBL1856519

SCHEMBL1856519

CCOC(=O)c1cccc(-c2cccc3c(F)c(Cc4cccc(C(F)(F)F)c4)sc23)c1.COCCNC(=O)c1cccc(-c2cccc3c(F)c(Cc4cccc(C(F)(F)F)c4)sc23)c1

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 18/20 0.65
MRGPRX4 Q96LA9 1/20 0.43
ALDH1A1 P00352 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3210910 0.95 GPR52 (0.71) GPR52MRGPRX4
SCHEMBL1855487 0.91 GPR52 (0.55) GPR52MRGPRX4ALDH1A1
SCHEMBL1849132 0.91 GPR52 (0.49) GPR52ALDH1A1
SCHEMBL1855818 0.90 GPR52 (0.65) GPR52MRGPRX4ALDH1A1POLB
SCHEMBL3211211 0.88 GPR52 (0.71) GPR52MRGPRX4
SCHEMBL3221538 0.87 GPR52 (0.60) GPR52MRGPRX4
SCHEMBL1851970 0.85 GPR52 (0.67) GPR52MRGPRX4
SCHEMBL1850978 0.83 GPR52 (0.49) GPR52ALDH1A1
SCHEMBL3209814 0.83 GPR52 (0.57) GPR52ALDH1A1POLB
SCHEMBL1848431 0.82 GPR52 (0.42) GPR52ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed