SCHEMBL18567883

SCHEMBL18567883

CC1(C)OB(c2cccc(/C(O)=C/C=N)c2)OC1(C)C

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P4HB P07237 1/20 0.42
LIPG Q9Y5X9 11/20 0.42
LPL P06858 10/20 0.42
IRAK4 Q9NWZ3 1/20 0.35
F11 P03951 2/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
ROCK1 Q13464 1/20 0.31
F2 P00734 1/20 0.31
PRSS1 P07477 1/20 0.31
PRSS2 P07478 1/20 0.31
PRSS3 P35030 1/20 0.31
FFAR1 O14842 1/20 0.31
EGFR P00533 1/20 0.31
PDGFRB P09619 1/20 0.30
KDR P35968 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30015761 0.77 P4HB (0.50) P4HBLIPGLPLF11CA1
SCHEMBL488896 0.77 P4HB (0.50) P4HBLIPGLPLF11CA1
SCHEMBL20894722 0.77 LIPG (0.50) P4HBLIPGLPLIRAK4F11
SCHEMBL14760399 0.77 LIPG (0.49) P4HBLIPGLPLIRAK4F11
SCHEMBL18567448 0.76 LIPG (0.41) P4HBLIPGLPLIRAK4F11
SCHEMBL4658432 0.75 L3MBTL1 (0.52) P4HBLIPGLPL
SCHEMBL30896588 0.75 L3MBTL1 (0.52) P4HBLIPGLPL
SCHEMBL23031277 0.74 LIPG (0.47) P4HBLIPGLPLIRAK4F11
SCHEMBL4782167 0.74 P4HB (0.47) P4HBLIPGLPLCA1CA2
SCHEMBL1476213 0.74 LIPG (0.59) P4HBLIPGLPLIRAK4F11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697210-B1 5-SUBSTITUTED IMINOTHIAZINES AND THEIR MONO-AND DIOXIDES AS BACE INHIBITORS, COMPOSITIONS, AND THEIR USE MERCK SHARP & DOHME (US) 2017-03-01 EP disclosed