SCHEMBL18567976

SCHEMBL18567976

C=C(c1ccccc1)c1ccc2c(c1)C1(c3ccccc3-2)c2ccccc2-c2ccc(C(=O)c3ccccc3)cc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 9/20 0.57
PTPRC P08575 1/20 0.43
TDP1 Q9NUW8 2/20 0.43
ATM Q13315 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 1/20 0.40
RARA P10276 1/20 0.40
RARB P10826 1/20 0.40
RARG P13631 1/20 0.40
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
RXRG P48443 1/20 0.40
CYP2C8 P10632 1/20 0.40
CYP2C9 P11712 1/20 0.40
SRD5A2 P31213 1/20 0.40
CNR2 P34972 1/20 0.39
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18900537 0.94 PDK2 (0.51) PDK2PTPRCTDP1RARARARB
SCHEMBL133477 0.91 PDK2 (0.66) PDK2PTPRCTDP1ATML3MBTL1
SCHEMBL1552743 0.91 PDK2 (0.66) PDK2PTPRCTDP1ATML3MBTL1
SCHEMBL16313987 0.91 PDK2 (0.47) PDK2PTPRCL3MBTL1ALDH1A1RARA
SCHEMBL12337045 0.88 PDK2 (0.60) PDK2PTPRCTDP1ATML3MBTL1
SCHEMBL134286 0.86 PDK2 (0.58) PDK2TDP1ATML3MBTL1THRB
SCHEMBL134285 0.86 PDK2 (0.58) PDK2TDP1ATML3MBTL1THRB
SCHEMBL29114 0.86 PDK2 (0.58) PDK2TDP1ATML3MBTL1THRB
SCHEMBL13702055 0.85 PDK2 (0.57) PDK2PTPRCTDP1ATML3MBTL1
SCHEMBL13702054 0.83 PDK2 (0.55) PDK2TDP1ATML3MBTL1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888706-B1 ORGANIC ELECTROLUMINESCENT DEVICE AND BORIC ACID AND BORINIC ACID DERIVATIVES USED THEREIN MERCK PATENT GMBH (DE) 2017-03-01 EP disclosed