SCHEMBL18569709

SCHEMBL18569709

Cc1ccnc(C(=O)N(CCO)CCO)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
MAPT P10636 1/20 0.49
HPGD P15428 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
TRPV1 Q8NER1 2/20 0.38
CTSA P10619 2/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
TP53 P04637 1/20 0.38
PKM P14618 1/20 0.38
UHRF1 Q96T88 1/20 0.37
CCR1 P32246 1/20 0.37
CCR5 P51681 1/20 0.37
CCR8 P51685 1/20 0.37
SSTR4 P31391 1/20 0.37
KDM4E B2RXH2 5/20 0.37
HSD17B10 Q99714 1/20 0.37
MEN1 O00255 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17297335 0.86 ALDH1A1 (0.41) ALDH1A1L3MBTL1MAPTCTSANPC1
SCHEMBL12677912 0.83 ALDH1A1 (0.69) ALDH1A1L3MBTL1MAPTHPGDTDP1
SCHEMBL6615353 0.81 ALDH1A1 (0.45) ALDH1A1L3MBTL1MAPTTRPV1NPC1
SCHEMBL4947098 0.78 ALDH1A1 (0.44) ALDH1A1L3MBTL1MAPTHPGDCTSA
SCHEMBL2160637 0.78 ALDH1A1 (0.44) ALDH1A1L3MBTL1MAPTCTSANPC1
SCHEMBL3677823 0.75 CES2 (0.52) ALDH1A1L3MBTL1HPGDSMN1; SMN2KDM4E
SCHEMBL16569986 0.74 ALDH1A1 (0.53) ALDH1A1L3MBTL1MAPTHPGDTDP1
SCHEMBL17820448 0.74 UHRF1 (0.43) ALDH1A1MAPTCTSANPC1RAB9A
SCHEMBL6985934 0.74 MAPT (0.43) ALDH1A1L3MBTL1MAPTHPGDTDP1
SCHEMBL13852609 0.72 KMT2A (0.52) CTSASMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2991981-B1 DIAMINOPYRAZINE COMPOUNDS, MEDICAMENTS CONTAINING SAID COMPOUNDS, USE THEREOF AND PROCESSES FOR THE PREPARATION THEREOF BOEHRINGER INGELHEIM INT (DE) 2017-03-01 EP disclosed