SCHEMBL18569864

SCHEMBL18569864

COC(=O)C(Cc1ccc(CCc2ccc(C(=O)O)cc2)cc1)NC(=O)CN(C)C(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.46
MDM4 O15151 1/20 0.43
MDM2 Q00987 1/20 0.43
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
KMT2A Q03164 1/20 0.41
HDAC1 Q13547 6/20 0.41
HDAC6 Q9UBN7 6/20 0.41
LNPEP Q9UIQ6 1/20 0.41
YAP1 P46937 1/20 0.40
OPRK1 P41145 1/20 0.39
GAA P10253 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18569502 0.91 NOS2 (0.44) KLK5MDM4MDM2HDAC1HDAC6
SCHEMBL2585645 0.86 MDM4 (0.55) KLK5MDM4MDM2ALDH1A1MEN1
SCHEMBL2585648 0.86 MDM4 (0.55) KLK5MDM4MDM2ALDH1A1MEN1
SCHEMBL16998490 0.83 ALDH1A1 (0.44) KLK5MDM4MDM2ALDH1A1LMNA
SCHEMBL15565791 0.83 ALDH1A1 (0.44) KLK5MDM4MDM2ALDH1A1LMNA
SCHEMBL15565793 0.83 ALDH1A1 (0.44) KLK5MDM4MDM2ALDH1A1LMNA
SCHEMBL18569863 0.81 KLK5 (0.44) KLK5MDM4MDM2ALDH1A1MEN1
SCHEMBL2583014 0.79 TACR1 (0.51) KLK5ALDH1A1YAP1
SCHEMBL2583010 0.79 TACR1 (0.51) KLK5ALDH1A1YAP1
SCHEMBL2792410 0.79 KLK5 (0.58) KLK5GAARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2882740-B1 IAP ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2017-03-01 EP disclosed