SCHEMBL2585645

SCHEMBL2585645

COC(=O)C(Cc1ccc(O)cc1)NC(=O)CN(C)C(=O)OC(C)(C)C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MDM4 O15151 1/20 0.55
MDM2 Q00987 1/20 0.55
LNPEP Q9UIQ6 3/20 0.49
NLRP3 Q96P20 1/20 0.48
KLK5 Q9Y337 1/20 0.47
NPSR1 Q6W5P4 2/20 0.47
KMT2A Q03164 2/20 0.47
ALDH1A1 P00352 2/20 0.47
TSHR P16473 1/20 0.47
CTSS P25774 1/20 0.46
CTSK P43235 1/20 0.46
LY96 Q9Y6Y9 1/20 0.44
KDR P35968 1/20 0.44
HDAC1 Q13547 2/20 0.43
HDAC6 Q9UBN7 2/20 0.43
ESR1 P03372 1/20 0.43
ESR2 Q92731 1/20 0.43
YAP1 P46937 1/20 0.43
MEN1 O00255 1/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2585648 1.00 MDM4 (0.55) MDM4MDM2LNPEPNLRP3KLK5
SCHEMBL2583065 0.89 CTSS (0.46) MDM4MDM2LNPEPCTSSCTSK
SCHEMBL2583067 0.89 CTSS (0.46) MDM4MDM2LNPEPCTSSCTSK
SCHEMBL18569864 0.86 KLK5 (0.46) MDM4MDM2LNPEPKLK5KMT2A
SCHEMBL18569863 0.84 KLK5 (0.44) MDM4MDM2KLK5KMT2AALDH1A1
SCHEMBL18569502 0.84 NOS2 (0.44) MDM4MDM2KLK5HDAC1HDAC6
SCHEMBL2583010 0.83 TACR1 (0.51) KLK5ALDH1A1YAP1
SCHEMBL2583014 0.83 TACR1 (0.51) KLK5ALDH1A1YAP1
SCHEMBL15604840 0.81 TSHR (0.54) MDM4MDM2LNPEPNLRP3KLK5
SCHEMBL16991034 0.81 TSHR (0.54) MDM4MDM2LNPEPNLRP3KLK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8350077-B2 Amides of creatine, method of their preparation, and remedy possessing a neuroprotective activity VERTEX CLOSED JOINT STOCK COMPANY (RU) 2013-01-08 US disclosed
US-20110269986-A1 AMIDES OF CREATNE, METHOD OF THEIR PREPARATION, AND REMEDY POSSESSING A NEUROPROTECTIVE ACTIVITY AMIDE BEVERAGE COMPANY, LLC 2011-11-03 US disclosed