SCHEMBL185704

SCHEMBL185704

CN(C)CCCCC(=O)NC1CC1.O=C(O)NCc1ccc(Nc2ccccc2C(F)(F)F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FASN P49327 2/20 0.43
SIGMAR1 Q99720 1/20 0.40
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
PTK2 Q05397 1/20 0.38
POLB P06746 4/20 0.38
GAA P10253 2/20 0.38
CYP3A4 P08684 3/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
EPHX1 P07099 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CYP2D6 P10635 2/20 0.36
EPHX2 P34913 1/20 0.36
PKM P14618 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL186742 0.97 SIGMAR1 (0.41) FASNSIGMAR1PTK2POLBGAA
SCHEMBL186097 0.94 SIGMAR1 (0.42) SIGMAR1PTK2POLBGAACYP3A4
SCHEMBL185584 0.89 SIGMAR1 (0.43) SIGMAR1POLBGAACYP3A4CYP1A2
SCHEMBL185464 0.88 SIGMAR1 (0.43) SIGMAR1PTK2POLBGAAKMT2A
SCHEMBL185364 0.85 SIGMAR1 (0.45) SIGMAR1PTK2POLBGAAKMT2A
SCHEMBL186322 0.84 SIGMAR1 (0.45) SIGMAR1POLBGAAKMT2AMEN1
SCHEMBL185935 0.83 SIGMAR1 (0.43) SIGMAR1POLBGAAKMT2AMEN1
SCHEMBL185809 0.83 SIGMAR1 (0.45) SIGMAR1POLBGAAKMT2AMEN1
SCHEMBL2808485 0.81 ALDH1A1 (0.38) POLBGAACYP3A4CYP1A2CYP2C9
SCHEMBL185673 0.81 POLB (0.45) SIGMAR1POLBGAACYP2C9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed
EP-2401256-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-01-04 EP disclosed
WO-2010097372-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed