SCHEMBL185926

SCHEMBL185926

O=C(O)Oc1ccnnc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.48
HSD17B10 Q99714 2/20 0.42
HDAC4 P56524 2/20 0.33
TBXA2R P21731 4/20 0.33
TBXAS1 P24557 3/20 0.33
LOXL2 Q9Y4K0 1/20 0.31
KMT2A Q03164 3/20 0.31
ALOX15 P16050 1/20 0.31
CYP19A1 P11511 1/20 0.31
ELANE P08246 1/20 0.31
LMNA P02545 1/20 0.30
MEN1 O00255 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27972799 0.85 LMNA (0.47) HCAR2HSD17B10KMT2AELANELMNA
SCHEMBL27950383 0.81 HCAR2 (0.42) HCAR2HSD17B10LOXL2KMT2AALOX15
SCHEMBL6628850 0.81 HCAR2 (0.42) HCAR2HSD17B10LOXL2KMT2AALOX15
SCHEMBL27455859 0.79 KMT2A (0.50) HCAR2HSD17B10KMT2AALOX15LMNA
SCHEMBL380364 0.75 HSD17B10 (0.56) HSD17B10KMT2ACYP19A1LMNAMEN1
SCHEMBL27950400 0.72 HCAR2 (0.33) HCAR2HSD17B10LOXL2
SCHEMBL31123876 0.72 KMT2A (0.56) HCAR2HSD17B10KMT2AALOX15LMNA
SCHEMBL876393 0.72 KMT2A (0.56) HCAR2HSD17B10KMT2AALOX15LMNA
SCHEMBL27672030 0.72
SCHEMBL465132 0.70 LMNA (0.52) HSD17B10KMT2AELANELMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0743574-B1 Migration imaging members XEROX CORP (US) 2000-12-27 EP claimed
EP-0743573-B1 Method for obtaining image contrast migration imaging members XEROX CORP (US) 2000-09-06 EP claimed
EP-0673783-B1 Recording sheets containing purine, pyrimidine, benzimidazole, imidazolidine, urazole, pyrazole, triazole, benzotriazole, tetrazole, and pyrazine compounds XEROX CORP (US) 2000-07-05 EP claimed
EP-2999338-B1 KNOWN AND NOVEL HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2017-07-12 EP disclosed
EP-2999338-A1 KNOWN AND NEW HETEROCYCLIC COMPOUNDS AS PEST CONTROL AGENTS Bayer CropScience Aktiengesellschaft (DE) 2016-03-30 EP disclosed
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed
EP-2401256-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-01-04 EP disclosed
WO-2010097372-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed
EP-1551830-B1 HETEROCYCLICALLY SUBSTITUTED INDOLINONES AND THEIR USE AS RECEPTOR TYROSINE KINASE INHIBATORS BOEHRINGER INGELHEIM PHARMA (DE) 2009-04-08 EP disclosed
EP-1551830-A2 HETEROCYCLICALLY SUBSTITUTED INDOLINONES AND THEIR USE AS RECEPTOR TYROSINE KINASE INHIBATORS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2005-07-13 EP disclosed
WO-2004026829-A2 HETEROCYCLICALLY SUBSTITUTED INDOLINONES AND THEIR USE AS RECEPTOR TYROSINE KINASE INHIBITORS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2004-04-01 WO disclosed
EP-0334289-B1 HETEROCYCLIC SUBSTITUTED 5,7-DIHYDROPYRROLO (3,2-F) BENZOXAZOL-6-ONES, PROCESS FOR THEIR PREPARATION AND DRUGS CONTAINING SAME Roche Diagnostics GmbH (DE) 1993-06-16 EP disclosed
EP-0334289-A1 Heterocyclic substituted 5,7-dihydropyrrolo (3,2-f) benzoxazol-6-ones, process for their preparation and drugs containing same Roche Diagnostics GmbH (DE) 1989-09-27 EP disclosed
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed