SCHEMBL18596299

SCHEMBL18596299

CCOCNc1ccc(Cl)cc1C(=O)NC/C=C/C(=O)OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.42
HPGD P15428 6/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
ALDH1A1 P00352 4/20 0.39
MAPT P10636 2/20 0.39
HSD17B10 Q99714 1/20 0.39
POLB P06746 3/20 0.38
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
MRGPRX1 Q96LB2 1/20 0.36
THRB P10828 1/20 0.36
RECQL P46063 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
KDM4E B2RXH2 1/20 0.35
CTSL P07711 2/20 0.35
CTSB P07858 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17447412 0.82 HSD17B10 (0.52) LMNAHPGDCYP1A2CYP3A4CYP2C19
SCHEMBL17445846 0.75 STAT3 (0.46) LMNAHPGDCYP1A2CYP3A4CYP2C19
SCHEMBL3354607 0.69 POLB (0.49) LMNAHPGDCYP1A2CYP2C19ALDH1A1
SCHEMBL3354613 0.69 POLB (0.49) LMNAHPGDCYP1A2CYP2C19ALDH1A1
SCHEMBL17447423 0.68 MEN1 (0.50) LMNAHPGDALDH1A1MAPTTDP1
SCHEMBL17447388 0.68 ALOX5 (0.41) LMNAHPGDALDH1A1MAPTHSD17B10
SCHEMBL17445812 0.68 MAOB (0.52) LMNAALDH1A1MAPTTDP1MEN1
SCHEMBL7310914 0.66 ALDH1A1 (0.50) LMNAHPGDALDH1A1MAPTPOLB
SCHEMBL7310907 0.66 ALDH1A1 (0.50) LMNAHPGDALDH1A1MAPTPOLB
SCHEMBL17445830 0.65 ALDH1A1 (0.57) HPGDCYP1A2CYP3A4CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9586890-B2 Screening methods for the binding affinity of chemical entities to biological molecules and NEDD4-1 inhibitors identified by the screening methods NORTHWESTERN UNIVERSITY (US) 2017-03-07 US disclosed