SCHEMBL18598680

SCHEMBL18598680

C[S+]([O-])Nc1ccc(N)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.39
ALDH1A1 P00352 4/20 0.39
CYP2C19 P33261 3/20 0.39
CYP3A4 P08684 3/20 0.39
HTT P42858 2/20 0.39
CYP1A2 P05177 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
CYP2C9 P11712 1/20 0.39
ALOX12 P18054 1/20 0.39
NR4A1 P22736 1/20 0.39
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
RAB9A P51151 2/20 0.38
RAD52 P43351 1/20 0.37
PKM P14618 2/20 0.36
ACHE P22303 1/20 0.36
TP53 P04637 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
KDM4E B2RXH2 1/20 0.34
APP P05067 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15947882 0.78 MAPT (0.41) MAPTALDH1A1CYP2C19CYP3A4HTT
SCHEMBL13148707 0.78 MAPT (0.42) MAPTALDH1A1CYP2C19CYP3A4HTT
SCHEMBL8010484 0.77 ALDH1A1 (0.43) MAPTALDH1A1L3MBTL1CYP2C9MEN1
SCHEMBL8009795 0.76 CA1 (0.35) APPCA1CA2CA9CA12
SCHEMBL13366567 0.76 CYP2A6 (0.38) MAPTALDH1A1CYP2C19CYP3A4HTT
Dimethyl Sulfoxide SCHEMBL18894360 0.76 MEN1 (0.57) MAPTALDH1A1CYP3A4L3MBTL1CYP2C9
SCHEMBL7294193 0.75 TSHR (0.43) MAPTALDH1A1CYP2C19CYP3A4CYP1A2
SCHEMBL18856695 0.74 MEN1 (0.48) MAPTALDH1A1CYP3A4NR4A1MEN1
SCHEMBL3723687 0.71
SCHEMBL14432373 0.71 ACHE (0.48) MAPTALDH1A1CYP2C19CYP3A4HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3705481-A1 HETEROARYL AMIDE COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITIONS THEREOF, AND APPLICATIONS THEREOF Rui Jin Hospital Affiliated To Shanghai Jiao Tong University School of Medicine (CN) 2020-09-09 EP disclosed
EP-2038286-B1 PYRRO[1,2-B]PYRIDAZINONE COMPOUNDS ANADYS PHARMACEUTICALS INC (US) 2017-03-08 EP disclosed